Polyaromatic heterocycles through intramolecular alkyne carbonyl metathesis: 5-Acylnaphtho[2,1-b]benzofurans

Maloy Nayak; Dileep Kumar Singh; Ikyon Kim

doi:10.1016/j.tet.2017.02.036

Polyaromatic heterocycles through intramolecular alkyne carbonyl metathesis: 5-Acylnaphtho[2,1-b]benzofurans

Maloy Nayak, Dileep Kumar Singh, Ikyon Kim

Department of Pharmacy

Research output: Contribution to journal › Article › peer-review

10 Citations (Scopus)

Abstract

A modular approach to 5-acylated naphtho[2,1-b]benzofurans was developed where Sonogashira cross-coupling and intramolecular alkyne carbonyl metathesis were sequentially employed to build the aromatic benzene C ring of naphtho[2,1-b]benzofuran with an acyl group at the C5 position.

Original language	English
Pages (from-to)	1831-1840
Number of pages	10
Journal	Tetrahedron
Volume	73
Issue number	14
DOIs	https://doi.org/10.1016/j.tet.2017.02.036
Publication status	Published - 2017

Bibliographical note

Funding Information:
This work was supported by the National Research Foundation of Korea grant funded by the Korea government (MSIP) (2014R1A2A1A11050491).

Publisher Copyright:
© 2017 Elsevier Ltd

All Science Journal Classification (ASJC) codes

Biochemistry
Drug Discovery
Organic Chemistry

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10.1016/j.tet.2017.02.036

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abstract = "A modular approach to 5-acylated naphtho[2,1-b]benzofurans was developed where Sonogashira cross-coupling and intramolecular alkyne carbonyl metathesis were sequentially employed to build the aromatic benzene C ring of naphtho[2,1-b]benzofuran with an acyl group at the C5 position.",

author = "Maloy Nayak and Singh, {Dileep Kumar} and Ikyon Kim",

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AU - Nayak, Maloy

AU - Singh, Dileep Kumar

AU - Kim, Ikyon

N1 - Funding Information: This work was supported by the National Research Foundation of Korea grant funded by the Korea government (MSIP) (2014R1A2A1A11050491). Publisher Copyright: © 2017 Elsevier Ltd

PY - 2017

Y1 - 2017

N2 - A modular approach to 5-acylated naphtho[2,1-b]benzofurans was developed where Sonogashira cross-coupling and intramolecular alkyne carbonyl metathesis were sequentially employed to build the aromatic benzene C ring of naphtho[2,1-b]benzofuran with an acyl group at the C5 position.

AB - A modular approach to 5-acylated naphtho[2,1-b]benzofurans was developed where Sonogashira cross-coupling and intramolecular alkyne carbonyl metathesis were sequentially employed to build the aromatic benzene C ring of naphtho[2,1-b]benzofuran with an acyl group at the C5 position.

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Polyaromatic heterocycles through intramolecular alkyne carbonyl metathesis: 5-Acylnaphtho[2,1-b]benzofurans

Abstract

Bibliographical note

All Science Journal Classification (ASJC) codes

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