Indium-catalyzed N -formylation of amines under solvent-free conditions

Joong Gon Kim; Doo Ok Jang

doi:10.1055/s-0029-1219784

Indium-catalyzed N -formylation of amines under solvent-free conditions

Joong Gon Kim, Doo Ok Jang

Chemistry and Medical Chemistry

Research output: Contribution to journal › Article › peer-review

51 Citations (Scopus)

Abstract

We have developed a simple, mild method for N-formylation of a wide variety of amines in the presence of indium metal as a catalyst under solvent-free conditions. This reaction is applicable to the chemoselective N-formylation of amino groups and -amino acid esters without epimerization.

Original language	English
Article number	U00810ST
Pages (from-to)	1231-1234
Number of pages	4
Journal	Synlett
Issue number	8
DOIs	https://doi.org/10.1055/s-0029-1219784
Publication status	Published - 2010

All Science Journal Classification (ASJC) codes

Organic Chemistry

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title = "Indium-catalyzed N -formylation of amines under solvent-free conditions",

abstract = "We have developed a simple, mild method for N-formylation of a wide variety of amines in the presence of indium metal as a catalyst under solvent-free conditions. This reaction is applicable to the chemoselective N-formylation of amino groups and -amino acid esters without epimerization.",

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AB - We have developed a simple, mild method for N-formylation of a wide variety of amines in the presence of indium metal as a catalyst under solvent-free conditions. This reaction is applicable to the chemoselective N-formylation of amino groups and -amino acid esters without epimerization.

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M1 - U00810ST

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Indium-catalyzed N -formylation of amines under solvent-free conditions

Abstract

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